Title:
Click chemistry inspired highly facile synthesis of triazolyl ethisterone glycoconjugates

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dc.contributor.authorDhananjay Kumar
dc.contributor.authorKunj B. Mishra
dc.contributor.authorBhuwan B. Mishra
dc.contributor.authorSaheli Mondal
dc.contributor.authorVinod K. Tiwari
dc.date.accessioned2026-02-07T06:00:48Z
dc.date.issued2014
dc.description.abstractNumerous deoxy-azido sugars 3 were prepared by the reaction of tosyl/bromo sugars with NaN3 in dry DMF under heating condition. The 1,3-dipolar cycloaddition of deoxy-azido sugars 3 with ethisterone 4 to afford regioselective triazole-linked ethisterone glycoconjugates 5 was investigated in the presence of CuI and DIPEA in dichloromethane or CuSO4· 5H2O and sodium ascorbate in aqueous medium. All the developed compounds were characterized by spectroscopic analysis (IR, 1H & 13C NMR, and MS spectra). Structure of triazolyl ethisterone glycoconjugate 5a has been further confirmed by its Single Crystal X-ray analysis. © 2013 Elsevier Inc. All rights reserved.
dc.identifier.doi10.1016/j.steroids.2013.11.022
dc.identifier.issn18785867
dc.identifier.urihttps://doi.org/10.1016/j.steroids.2013.11.022
dc.identifier.urihttps://dl.bhu.ac.in/bhuir/handle/123456789/26353
dc.subjectCarbohydrate
dc.subjectClick chemistry
dc.subjectEthisterone
dc.subjectGlycoconjugate
dc.titleClick chemistry inspired highly facile synthesis of triazolyl ethisterone glycoconjugates
dc.typePublication
dspace.entity.typeArticle

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